Contents
The Medicinal Chemist's Guide to Solving ADMET Challenges
Drug Discovery Series
Editor-in-chief
David Thurston, King's College London, UK
Series editors:
David Fox, Vulpine Science and Learning, UK
Ana Martinez, Centro de Investigaciones Biologicas-CSIC, Spain
Hong Shen, Roche Innovation Center Shanghai, China
Ian Storer, AstraZeneca, UK
Editorial advisor:
Corey Hopkins, University of Nebraska Medical Center, USA
Titles in the Series:
1: Metabolism, Pharmacokinetics and Toxicity of Functional Groups
2: Emerging Drugs and Targets for Alzheimer's Disease; Volume 1
3: Emerging Drugs and Targets for Alzheimer's Disease; Volume 2
4: Accounts in Drug Discovery
5: New Frontiers in Chemical Biology
6: Animal Models for Neurodegenerative Disease
7: Neurodegeneration
8: G Protein-Coupled Receptors
9: Pharmaceutical Process Development
10: Extracellular and Intracellular Signaling
11: New Synthetic Technologies in Medicinal Chemistry
12: New Horizons in Predictive Toxicology
13: Drug Design Strategies: Quantitative Approaches
14: Neglected Diseases and Drug Discovery
15: Biomedical Imaging
16: Pharmaceutical Salts and Cocrystals
17: Polyamine Drug Discovery
18: Proteinases as Drug Targets
19: Kinase Drug Discovery
20: Drug Design Strategies: Computational Techniques and Applications
21: Designing Multi-target Drugs
22: Nanostructured Biomaterials for Overcoming Biological Barriers
23: Physico-Chemical and Computational Approaches to Drug Discovery
24: Biomarkers for Traumatic Brain Injury
25: Drug Discovery from Natural Products
26: Anti-inflammatory Drug Discovery
27: New Therapeutic Strategies for Type 2 Diabetes: Small Molecules
28: Drug Discovery for Psychiatric Disorders
29: Organic Chemistry of Drug Degradation
30: Computational Approaches to Nuclear Receptors
31: Traditional Chinese Medicine
32: Successful Strategies for the Discovery of Antiviral Drugs
33: Comprehensive Biomarker Discovery and Validation for Clinical Application
34: Emerging Drugs and Targets for Parkinson's Disease
35: Pain Therapeutics; Current and Future Treatment Paradigms
36: Biotherapeutics: Recent Developments using Chemical and Molecular Biology
37: Inhibitors of Molecular Chaperones as Therapeutic Agents
38: Orphan Drugs and Rare Diseases
39: Ion Channel Drug Discovery
40: Macrocycles in Drug Discovery
41: Human-based Systems for Translational Research
42: Venoms to Drugs: Venom as a Source for the Development of Human Therapeutics
43: Carbohydrates in Drug Design and Discovery
44: Drug Discovery for Schizophrenia
45: Cardiovascular and Metabolic Disease: Scientific Discoveries and New Therapies
46: Green Chemistry Strategies for Drug Discovery
47: Fragment-based Drug Discovery
48: Epigenetics for Drug Discovery
49: New Horizons in Predictive Drug Metabolism and Pharmacokinetics
50: Privileged Scaffolds in Medicinal Chemistry: Design, Synthesis, Evaluation
51: Nanomedicines: Design, Delivery and Detection
52: Synthetic Methods in Drug Discovery: Volume 1
53: Synthetic Methods in Drug Discovery: Volume 2
54: Drug Transporters: Role and Importance in ADME and Drug Development
55: Drug Transporters: Recent Advances and Emerging Technologies
56: Allosterism in Drug Discovery
57: Anti-aging Drugs: From Basic Research to Clinical Practice
58: Antibiotic Drug Discovery: New Targets and Molecular Entities
59: Peptide-based Drug Discovery: Challenges and New Therapeutics
60: Drug Discovery for Leishmaniasis
61: Biophysical Techniques in Drug Discovery
62: Acute Brain Impairment Through Stroke: Drug Discovery and Translational Research
63: Theranostics and Image Guided Drug Delivery
64: Pharmaceutical Formulation: The Science and Technology of Dosage Forms
65: Small-molecule Transcription Factor Inhibitors in Oncology
66: Therapies for Retinal Degeneration: Targeting Common Processes
67: Kinase Drug Discovery: Modern Approaches
68: Advances in Nucleic Acid Therapeutics
69: MicroRNAs in Diseases and Disorders: Emerging Therapeutic Targets
70: Emerging Drugs and Targets for Multiple Sclerosis
71: Cytotoxic Payloads for AntibodyDrug Conjugates
72: Peptide Therapeutics: Strategy and Tactics for Chemistry, Manufacturing, and Controls
73: Anti-fibrotic Drug Discovery
74: Protein Degradation with New Chemical Modalities: Successful Strategies in Drug Discovery and Chemical Biology
75: Artificial Intelligence in Drug Discovery
76: New Tools to Interrogate Endocannabinoid Signalling: From Natural Compounds to Synthetic Drugs
77: Phenotypic Drug Discovery
78: ProteinProtein Interaction Regulators
79: The Medicinal Chemist's Guide to Solving ADMET Challenges
How to obtain future titles on publication:
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For further information please contact:
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The Medicinal Chemists Guide to Solving ADMET Challenges
Edited by
Patrick Schnider
Rejuveron Life Sciences AG, Switzerland
E-mail:
Drug Discovery Series No. 79
Print ISBN: 978-1-78801-227-0
PDF ISBN: 978-1-78801-641-4
EPUB ISBN: 978-1-83916-049-3
Print ISSN: 2041-3203
Electronic ISSN: 2041-3211
A catalogue record for this book is available from the British Library
The Royal Society of Chemistry
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